FGF R4

FGF R4 詳細

英語名Fibroblast growth factor receptor 4市販薬剤の数3
治験薬の数19ターゲットの別称CD334 Antigen,EC 2.7.10.1,FGFR-4,Receptor, Fibroblast Growth Factor, Type 4,EC 2.7.10,JTK2,Tyrosine Kinase Related To Fibroblast Growth Factor Receptor,Hydroxyaryl-Protein Kinase,Tyrosylprotein Kinase,EC:2.7.10.1,Fibroblast growth factor receptor 4,CD334,FGFR4,TKF
研究&開発段階Approved
英語名Fibroblast growth factor receptor 4
ターゲットの別称CD334 Antigen,EC 2.7.10.1,FGFR-4,Receptor, Fibroblast Growth Factor, Type 4,EC 2.7.10,JTK2,Tyrosine Kinase Related To Fibroblast Growth Factor Receptor,Hydroxyaryl-Protein Kinase,Tyrosylprotein Kinase,EC:2.7.10.1,Fibroblast growth factor receptor 4,CD334,FGFR4,TKF
市販薬剤の数3
治験薬の数19
研究&開発段階Approved

FGF R4 製品リスト

  • 属性

    Protein (2)

  • 製品ライブラリ

    オンライン (2)

  • Human (2)

  • タグ

    His Tag (1)Fc Tag (1)

  • マーカー

    Unconjugated (2)

製品番号発現システム製品説明タンパク質の構造純度特性
FG4-H5228
Human
HEK293
Human FGF R4 / CD334 Protein, His Tag, low endotoxin
FG4-H5253
Human
HEK293
Human FGF R4 / CD334 Protein, Fc Tag (MALS & SPR verified)
総数量2
  • 1

FGF R4バックグランド

Fibroblast growth factor receptor 4(FGFR4) is also known as CD334, JTK2, hydroxyaryl-protein kinase, TKF, protein-tyrosine kinase . The FGFR4 gene provides instructions for making a protein called fibroblast growth factor receptor 4. This protein is part of a family of fibroblast growth factor receptors that share similar structures and functions. These receptor proteins play a role in important processes such as cell division, regulating cell growth and maturation, formation of blood vessels, wound healing, and embryo development.The FGFR4 protein interacts with specific growth factors to conduct signals from the environment outside the cell to the nucleus. The nucleus responds to these signals by switching on or off appropriate genes that help the cell adjust to changes in the environment. In response, the cell might divide, move, or mature to take on specialized functions. Although specific functions of FGFR4 remain unclear, studies indicate that the gene is involved in muscle development and the maturation of bone cells in the skull. The FGFR4 gene may also play a role in the development and maintenance of specialized cells (called foveal cones) in the light-sensitive layer (the retina) at the back of the eye.

FGF R4分子の別称

FGFR4,CD334,JTK2,MGC20292,TKF

治験薬に関する情報

英語名研究コード研究開発ステージ会社適応症臨床試験
SC-0011SC-0011Phase 3 ClinicalShijiazhuang Zhikang Hongren New Drug Development Co LtdCarcinoma, Non-Small-Cell Lung; Esophageal Neoplasms; Gastroesophageal Junction Neoplasms; Solid tumours; Stomach Neoplasms
詳細
AUR-109ODM-203; AUR-109Phase 2 ClinicalOrion CorpBreast Neoplasms; Carcinoma, Renal Cell; Colorectal Neoplasms; Kidney Neoplasms; Liver Neoplasms; Lung Neoplasms; Ovarian Neoplasms; Pulmonary Fibrosis; Solid tumours; Urinary Bladder Neoplasms
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RogaratinibBAY-1163877Phase 2 ClinicalBayer AGBreast Neoplasms; Carcinoma, Non-Small-Cell Lung; Carcinoma, Transitional Cell; Gastrointestinal Stromal Tumors; Metastatic breast cancer; Neoplasms; Sarcoma; Solid tumours; Urinary Bladder Neoplasms
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FisogatinibBLU-554; CS-3008Phase 2 ClinicalBlueprint Medicines CorpCarcinoma, Hepatocellular
詳細
BB-102BB-102; BB102Phase 2 ClinicalBroadenbio Co LtdCarcinoma, Hepatocellular; Solid tumours
詳細
GunagratinibICP-192Phase 2 ClinicalBeijing Tiancheng Pharmaceutical Technology Co LtdBiliary Tract Neoplasms; Carcinoma, Transitional Cell; Cholangiocarcinoma; Head and Neck Neoplasms; Lung Neoplasms; Solid tumours; Stomach Neoplasms; Urinary Bladder Neoplasms
詳細
IrpagratinibABSK-011Phase 2 ClinicalABbisko Therapeutics Co LtdCarcinoma, Hepatocellular; Liver Neoplasms; Solid tumours
詳細
BPI-43487BPI-43487Phase 1 ClinicalBetta Pharmaceuticals Co LtdBiliary Tract Neoplasms; Carcinoma, Hepatocellular; Solid tumours
詳細
HS-236HS-236Phase 1 ClinicalZhejiang Hisun Pharmaceutical Co LtdSolid tumours
詳細
HS-10340HS-10340Phase 1 ClinicalChangzhou Hengbang Pharmaceutical Co Ltd, Jiangsu Hansoh Pharmaceutical Group Co Ltd, Shanghai Hansoh Biomedical Co LtdSolid tumours
詳細
ICP-105ICP-105Phase 1 ClinicalBeijing Innocare Pharma Tech Co Ltd, Beijing Tiancheng Pharmaceutical Technology Co Ltd, Nanjing Tianyin Jianhua Pharmaceutical Technology Co LtdLiver Neoplasms; Solid tumours
詳細
ZSP-1241ZSP-1241Phase 1 ClinicalGuangdong Zhongsheng Pharmaceutical Co Ltd, Wuxi Apptec Co LtdBiliary Tract Neoplasms; Carcinoma; Carcinoma, Hepatocellular; Cholangiocarcinoma; Colorectal Neoplasms; Esophageal Neoplasms; Liver Neoplasms; Stomach Neoplasms
詳細
H3B-6527H3B-6527Phase 1 ClinicalH3 Biomedicine IncCarcinoma, Hepatocellular; Liver Neoplasms
詳細
FGFR4-CAR T Cells Therapy(National Cancer Institute)Phase 1 ClinicalNational Cancer InstituteRhabdomyosarcoma
詳細
TYRA-430TYRA-430Phase 1 ClinicalTyra Biosciences IncCarcinoma, Hepatocellular; Neoplasms; Solid tumours
詳細
SYHX-2005SYHX-2005; SYHX2005Phase 1 ClinicalCspc Ouyi Pharmaceutical Co LtdSolid tumours
詳細
JAB-6343Phase 1 ClinicalJacobio Pharmaceuticals Co LtdSolid tumours
詳細
SY-4798SY-4798Phase 1 ClinicalShouyao Holding (Beijing) Co LtdBiliary Tract Neoplasms; Carcinoma, Hepatocellular; Solid tumours
詳細
ABSK-012ABSK-012; ABSK012Phase 1 ClinicalABbisko Therapeutics Co LtdSolid tumours
詳細

市販薬剤に関する情報

英語名研究コード研究開発ステージ会社オリジナル製品名最初に承認をした国最初の適応症最初に承認を受けた会社承認された日付適応症臨床試験
Lenvatinib MesilateE-7080; MK-7902; ER-203492-00ApprovedEisai Co LtdKisplyx, Lenvima, Lenvima/Kisplyx, 乐卫玛United StatesThyroid NeoplasmsEisai Inc2015-02-13Adenocarcinoma; Adenocarcinoma of Lung; Adenocarcinoma, Follicular; Biliary Tract Neoplasms; Breast Neoplasms; Carcinoma, Adenoid Cystic; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Renal Cell; Carcinoma, Squamous Cell; Cholangiocarcinoma; Endometrial Neoplasms; Esophageal Neoplasms; Gastrointestinal Stromal Tumors; Glioma; Hepatic Insufficiency; Liver Diseases; Liver Neoplasms; Lymphoma; Melanoma; Neoplasm Metastasis; Neoplasms; Neuroendocrine Tumors; Osteosarcoma; Ovarian Neoplasms; Paraganglioma; Pheochromocytoma; Renal Insufficiency; Solid tumours; Stomach Neoplasms; Thyroid Cancer, Papillary; Thyroid Carcinoma, Anaplastic; Thyroid Neoplasms; Uterine Cervical Neoplasms
詳細
FutibatinibTAS-120ApprovedOtsuka Pharmaceutical Co Ltd, Taiho Pharmaceutical Co LtdLYTGOBIUnited StatesCholangiocarcinomaTaiho Oncology Inc2022-09-30Biliary Tract Neoplasms; Bone Marrow Neoplasms; Breast Neoplasms; Carcinoma; Carcinoma, Non-Small-Cell Lung; Carcinoma, Transitional Cell; Central Nervous System Neoplasms; Cholangiocarcinoma; Endometrial Neoplasms; Esophageal Neoplasms; Lymphoma; Metastatic breast cancer; Neoplasm Metastasis; Neoplasms; Sarcoma; Solid tumours; Stomach Neoplasms
詳細
Erdafitinib890E37NHMV; G-024; JNJ-493; JNJ-42756493; TAR-210ApprovedAstex Pharmaceuticals IncBalversa, 博珂United StatesCarcinoma, Transitional CellJanssen Biotech Inc2019-04-12Adenocarcinoma; Bile Duct Neoplasms; Bone metastases; Carcinoma; Carcinoma, Hepatocellular; Carcinoma, Neuroendocrine; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Carcinoma, Transitional Cell; Central Nervous System Neoplasms; Ependymoma; Esophageal Neoplasms; Glioma; Hepatic Insufficiency; Hepatoblastoma; Histiocytic Sarcoma; Histiocytosis, Langerhans-Cell; Lymphoma; Lymphoma, Non-Hodgkin; Medulloblastoma; Metastatic breast cancer; Multiple Myeloma; Neoplasms; Neoplasms, Germ Cell and Embryonal; Neuroblastoma; Neuroectodermal Tumors, Primitive, Peripheral; Osteosarcoma; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Rhabdoid Tumor; Rhabdomyosarcoma; Sarcoma; Sarcoma, Ewing; Solid tumours; Stomach Neoplasms; Urinary Bladder Neoplasms; Urologic Neoplasms; Wilms Tumor; Xanthogranuloma, Juvenile
詳細
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